BDBM50525951 CHEMBL4447367

SMILES CC(C)[C@H]1CN(CCN1C)c1nc2cc(F)ccc2c(=O)n1-c1ccc(cc1)C(F)(F)F

InChI Key InChIKey=FPPDJHDANGQLEF-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50525951   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Asahi Kasei Medical

Curated by ChEMBL

LigandBDBM50525951(CHEMBL4447367)Copy SMILESCopy InChI

Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/25/2021
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