BDBM50525946 CHEMBL4586856

SMILES CN1CCN(CC1)c1nc2ccc(F)cc2c(=O)n1-c1ccc(OC(F)(F)F)cc1

InChI Key InChIKey=APUUNOKUBAGYKV-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50525946   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Asahi Kasei Medical

Curated by ChEMBL

LigandBDBM50525946(CHEMBL4586856)Copy SMILESCopy InChI

Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/25/2021
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