BDBM50525943 CHEMBL4449850

SMILES COc1ccc(cc1)-n1c(nc2cc(F)ccc2c1=O)N1CCN(C)CC1

InChI Key InChIKey=YKXWTUJCWBZVDN-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50525943   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Asahi Kasei Medical

Curated by ChEMBL

LigandBDBM50525943(CHEMBL4449850)Copy SMILESCopy InChI

Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/25/2021
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