BDBM50520957 CHEMBL4458265

SMILES Cc1cc(O)c(-c2ccc(cc2)C2(CN)CC2)c2c1[nH]c(=O)c1ccccc21

InChI Key InChIKey=AIOQBMZRABXSCF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50520957   

TargetLymphokine-activated killer T-cell-originated protein kinase(Human)
Sichuan University

Curated by ChEMBL

LigandBDBM50520957(CHEMBL4458265)Copy SMILESCopy InChI

Affinity DataIC50: 25nMAssay Description:Inhibition of human TOPK using MBP as substrate after 2 hrs in presence of [gamma-33P]-ATP by filter-binding methodMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL