BDBM50518422 CHEMBL4448100

SMILES Cc1cccc(Cl)c1NC(=O)C1(C)CC2c3ccccc3C1c1cc(Cl)ccc21

InChI Key

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50518422   

TargetD(1A) dopamine receptor(Rat)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50518422(CHEMBL4448100)
Affinity DataEC50:  332nMAssay Description:Positive allosteric modulation of rat D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulation relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50518422(CHEMBL4448100)
Affinity DataEC50:  22nMAssay Description:Positive allosteric modulation of human D1R expressed in HEK cells assessed as increase in dopamine-induced cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed