BDBM50517789 CHEMBL4518858

SMILES COc1ncc(cc1C)N1CCc2ncnc(Nc3cccc(c3)C(=O)NC3CCOCC3)c2C1

InChI Key InChIKey=XRSJOEAILRNBRZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50517789   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50517789(CHEMBL4518858)Copy SMILESCopy InChI

Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant human PI3Kdelta using PIP2 as substrate after 35 to 40 mins by HTRF assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/22/2021
Entry Details Article
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