BDBM50515337 CHEMBL4560240

SMILES COc1cc(\C=C\C(=O)NCCCCCCNC23CC4CC(C)(CC(C)(C4)C2)C3)ccc1O

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50515337   

TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Alma Mater Studiorum - University of Bologna

Curated by ChEMBL
LigandPNGBDBM50515337(CHEMBL4560240)
Affinity DataIC50: 6.90E+3nMAssay Description:Antagonist activity at GluN1a/GluN2A (unknown origin) expressed in Xenopus laevis oocytes at -60 mV holding potential by voltage clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
Alma Mater Studiorum - University of Bologna

Curated by ChEMBL
LigandPNGBDBM50515337(CHEMBL4560240)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of GluN1/GluN2B NMDA receptor (unknown origin) expressed in xenopus laevis oocytes with holding potential of -70 mV by two-electrode volta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed