BDBM50514006 CHEMBL4572843

SMILES Fc1ccc(cc1)C(CCCNCC1CCc2[nH]c3ccc(F)cc3c2C1)c1ccc(F)cc1

InChI Key InChIKey=OCZIMUMAPGQEBH-UHFFFAOYSA-N

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50514006   

LigandPNGBDBM50514006(CHEMBL4572843)
Affinity DataIC50: 710nMAssay Description:Inhibition of VPS4B (unknown origin) assessed as reduction in ATPase activity in presence of activating fragment of substrate CHMP1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514006(CHEMBL4572843)
Affinity DataIC50: 710nMAssay Description:Inhibition of VPS4B (unknown origin) by malachite green assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514006(CHEMBL4572843)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of p97 (unknown origin) by malachite green assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
LigandPNGBDBM50514006(CHEMBL4572843)
Affinity DataIC50: 710nMAssay Description:Inhibition of recombinant VPS4B (unknown origin) expressed in Escherichia coli (DE3) incubated for 10 mins by malachite green based ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
LigandPNGBDBM50514006(CHEMBL4572843)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of recombinant p97 (unknown origin) expressed in Escherichia coli (DE3) incubated for 30 mins by malachite green based ATPase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed