BDBM50505549 CHEMBL4466785

SMILES OC[C@]1(O)CN(C[C@@H]1S(=O)(=O)c1ccc(cc1)C#N)S(=O)(=O)c1ccc(Cl)cn1

InChI Key InChIKey=ITJSJRXBFTUEAW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50505549   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50505549(CHEMBL4466785)Copy SMILESCopy InChI

Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at BacMam virus expressing human TRPV4 transduced in BHK/AC9 or HEK MSR2 cells assessed as inhibition of GSK634775-induced Ca2+ f...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/18/2021
Entry Details Article
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