BDBM50500495 CHEMBL3745992

SMILES Cc1cccc(C(=O)Nc2cc([nH]n2)-c2nc3ccccc3[nH]2)c1Cl

InChI Key InChIKey=MZSONBOADBXTJB-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50500495   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Astrazeneca

Curated by ChEMBL

LigandBDBM50500495(CHEMBL3745992)Copy SMILESCopy InChI

Affinity DataIC50: 280nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 2 hrs by FRET a...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
9/4/2020
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