BDBM50498117 CHEMBL3403044

SMILES CCn1cc(NC(=O)c2ccc(Cn3nc(C)c(Br)c3C)o2)c(n1)C(N)=O

InChI Key InChIKey=ZIIPBQJCNHJSMA-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50498117   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL

LigandBDBM50498117(CHEMBL3403044)Copy SMILESCopy InChI

Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of HIF1 in human HT1080 cells transfected with 5xHRE/pGL3/VEGF/E1b reporter plasmid pre-incubated for 1 hr followed by incubation under hy...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In Depth
Date in BDB:
9/3/2020
Entry Details Article
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