BDBM50484551 CHEMBL1933928

SMILES CC1(C)CNC(=O)c2sc(Nc3ccc(I)cc3Cl)c(C(=O)NOC[C@H](O)CO)c2C1

InChI Key InChIKey=NUTGQSGXRGUYMD-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50484551   

TargetDual specificity mitogen-activated protein kinase kinase 1/2(Human)
Ucb Pharma

Curated by ChEMBL

LigandBDBM50484551(CHEMBL1933928)Copy SMILESCopy InChI

Affinity DataIC50: 9nMAssay Description:Inhibition of human MEK using fluorescein-labelled Erk-tide as substrate after 20 mins by IMAP assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/29/2020
Entry Details Article
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