BDBM50484272 CHEMBL1824131

SMILES COc1ccc(cc1OC)S(=O)(=O)N(CC(C)C)Cc1ccc2OC(C)(C)C=Cc2c1

InChI Key InChIKey=XNFHNRBWLZQXJI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50484272   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Emory University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50484272(CHEMBL1824131)
Affinity DataIC50: 672nMAssay Description:Inhibition of hypoxia-induced HIF1 activation in human LN229 cells expressing HRE-AP reporter gene preincubated for 1 hr under normoxia condition fol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed