BDBM50479921 CHEMBL508166

SMILES CS\C=C(\C)n1c(noc1=O)C(=O)c1ccc(Br)cc1

InChI Key InChIKey=DDTZWTBRUYDWQL-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50479921   

TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50479921(CHEMBL508166)
Affinity DataIC50: 2.52E+4nMAssay Description:Inhibition of L-type calcium channel in Wistar rat tail artery smooth muscle cells assessed as blockade of barium-sensitive inward rectifying current...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Universita Degli Studi Di Bologna

Curated by ChEMBL
LigandPNGBDBM50479921(CHEMBL508166)
Affinity DataKi:  490nMAssay Description:Displacement of [3H]diltiazem from L-type calcium channel in Sprague-Dawley rat cardiac myocytes by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed