BDBM50471064 CHEMBL301810

SMILES OC(=O)c1cc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2cc3ccccc3cc2C(=O)NCC23CC4CC(CC(C4)C2)C3)cc(c1)C(O)=O

InChI Key

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50471064   

TargetGastrin/cholecystokinin type B receptor(Mouse)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)
Affinity DataKi:  13nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to mouse cortical membrane Cholecystokinin 2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)
Affinity DataKi:  13nMAssay Description:In vitro inhibitory activity against Cholecystokinin type B receptor using [125I]BH-CCK-8S as radioligand in mouse cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)
Affinity DataKi:  794nMAssay Description:Inhibition of 20 pM [125I]BH-CCK-8S binding to guinea pig pancreas membrane Cholecystokinin 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)
Affinity DataKi:  794nMAssay Description:Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50471064(CHEMBL301810)
Affinity DataKi:  851nMAssay Description:In vitro inhibitory activity against Cholecystokinin type A receptor using [125I]BH-CCK-8S as radioligand in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed