BDBM50470617 CHEMBL137180

SMILES OC(=O)c1cc(NC(=O)[C@H](Cc2ccccc2)NC(=O)C2C(C3c4ccccc4C2c2ccccc32)C(=O)NCc2ccc3ccccc3c2)cc(c1)C(O)=O

InChI Key

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50470617   

TargetGastrin/cholecystokinin type B receptor(Mouse)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50470617(CHEMBL137180)
Affinity DataKi:  2.70nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S for Cholecystokinin type B receptor binding sites in mouse cortical homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50470617(CHEMBL137180)
Affinity DataKi:  1.62E+3nMAssay Description:Competition with 20 pM [125I]BH-CCK-8S at Cholecystokinin type A receptor binding sites on guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed