BDBM50469175 CHEMBL4282148
SMILES CCOC(=O)C1CCN(CC1)c1ccc2c(Nc3cc(C)[nH]n3)nc(nc2c1)-c1ccccc1
InChI Key InChIKey=JYWBPBWVUMVNAE-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50469175
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells at -80 mV holding potential by whole-cell patch clamp methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.52E+3nMAssay Description:Inhibition of Aurora B (unknown origin) using FAM-labelled peptide as substrate pretreated for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of Aurora A (unknown origin) using FAM-labelled peptide as substrate pretreated for 10 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair