BDBM50467932 CHEMBL4294577

SMILES COc1cc2CCN(CCCCNC(=O)c3ccc(F)cc3)Cc2cc1O

InChI Key InChIKey=QOEWXLMSFYFGOV-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50467932   

TargetD(3) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50467932(CHEMBL4294577)
Affinity DataEC50:  490nMAssay Description:Antagonist activity at human dopamine D3 receptor assessed as inhibition of beta-arrestin recruitment by Tango assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50467932(CHEMBL4294577)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D3 receptor expressed in HEKT cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
City University of New York

Curated by ChEMBL
LigandPNGBDBM50467932(CHEMBL4294577)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]N-Methylspiperone from human dopamine D4 receptor expressed in HEK cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed