BDBM50466571 CHEMBL4278148

SMILES Cn1c2ccc(cc2c(=O)n(Cc2cnc[nH]2)c1=O)S(=O)(=O)NC1(C)CC1

InChI Key InChIKey=YXPICKMFLQULDH-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50466571   

TargetPoly(ADP-ribose) glycohydrolase(Human)
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50466571(CHEMBL4278148)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of human full length PARG using Bt-NAD ribosylated PARP1 substrate after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed