BDBM50465937 CHEMBL4287192

SMILES Cc1cc(Oc2nccc3occc23)ccc1-c1cncc2ncnn12

InChI Key InChIKey=OUGRRYAUMLQMJR-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50465937   

TargetD(1A) dopamine receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50465937(CHEMBL4287192)
Affinity DataEC50:  5.49E+3nMAssay Description:Agonist activity at human dopamine D1 receptor expressed in HEK293T cells assessed as induction of cAMP levels after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50465937(CHEMBL4287192)
Affinity DataKi:  2.35E+3nMAssay Description:Displacement of [3H]-SCH23390 from human dopamine D1 receptor expressed in LTK cell membranes after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed