BDBM50463966 CHEBI:28822::Elcosanoic Acid

SMILES CCCCCCCCCCCCCCCCCCCC(=O)O

InChI Key InChIKey=VKOBVWXKNCXXDE-UHFFFAOYSA-N

Data  7 IC50

PDB links: 7 PDB IDs match this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50463966   

TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Martin-Luther-University Halle-Wittenberg

Curated by ChEMBL
LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 20 mins followed by substrate addition and measured at 1...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]GW2331 from Homo sapiens (human) PPARalpha receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article

LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]BRL49653 from Homo sapiens (human) PPARgamma receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article

LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]GW2433 from Homo sapiens (human) PPARdelta receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article

TargetTyrosine-protein phosphatase non-receptor type 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50463966(CHEBI:28822 | Elcosanoic Acid)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of PTP1B (unknown origin) using pNPP as substrate incubated for 30 mins by photometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed