BDBM50463897 CHEMBL4241205

SMILES Cc1noc(C)c1-c1cc(N)c2ncn(Cc3ccc(cc3)C3CO3)c2c1

InChI Key InChIKey=XINQCOMOQIYWTG-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50463897   

TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 4 hrs by alpha-screen as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 274nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 5 mins by alpha-screen a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1/BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-scr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 50nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 30 mins by alpha-screen ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Zenith Epigenetics

Curated by ChEMBL
LigandPNGBDBM50463897(CHEMBL4241205)
Affinity DataIC50: 75nMAssay Description:Inhibition of N-terminal His-tagged BRD4 (BD1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide after 1 hr by alpha-screen ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed