BDBM50454837 CHEMBL4217784

SMILES Clc1c2C(=O)N(C(=O)c2c(Cl)c(Cl)c1Cl)c1ccccc1\C=C\c1cccs1

InChI Key InChIKey=CSRGGIVFZAJPIC-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50454837   

TargetOxysterols receptor LXR-beta(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454837(CHEMBL4217784)
Affinity DataEC50:  559nMAssay Description:Agonist activity at human LXRbeta expressed in HEK293 cells co-expressing CMX-beta-galactosidase incubated for 16 hrs by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetOxysterols receptor LXR-beta(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454837(CHEMBL4217784)
Affinity DataEC50:  790nMAssay Description:Agonist activity at mouse LXRbeta expressed in HEK293 cells co-expressing CMX-beta-galactosidase incubated for 16 hrs by luciferase reporter gene ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetOxysterols receptor LXR-alpha(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50454837(CHEMBL4217784)
Affinity DataEC50:  40nMAssay Description:Agonist activity at LXRbeta ligand-binding domain (unknown origin) incubated for 1.5 hrs using fluorescein-labeled coactivator peptide by TR-FRET com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed