BDBM50442422 CHEMBL2443089

SMILES FC(F)(F)c1ccc(NC(=O)N2CCC3(CC2)CCc2cccc(Cl)c2O3)c(Cl)c1

InChI Key InChIKey=MDXKLWVCMQHWSJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442422   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Glenmark Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50442422(CHEMBL2443089)
Affinity DataIC50: 178nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed