BDBM50442419 CHEMBL2443066

SMILES Fc1ccc2nc(NC(=O)N3CCC4(CC3)CCc3cccc(Cl)c3O4)sc2c1

InChI Key InChIKey=TVHROQADBLZZQX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442419   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Glenmark Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50442419(CHEMBL2443066)
Affinity DataIC50: 113nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed