BDBM50442411 CHEMBL2443073

SMILES OC1CC2(CCN(CC2)C(=O)Nc2ccc(cc2)C(F)(F)F)Oc2c(Cl)cccc12

InChI Key InChIKey=IELJAKQICRQYBF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50442411   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Glenmark Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50442411(CHEMBL2443073)
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed