BDBM50432948 CHEMBL2377737

SMILES Cn1c(NC(=O)N(CCC(c2ccccc2)c2ccccc2)CCN2CCOCC2)nc2ccccc12

InChI Key InChIKey=FSQOBTYKZNGUPP-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50432948   

TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandPNGBDBM50432948(CHEMBL2377737)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR expressed in CHO cells assessed as increase in intracellular calcium level after 5 hrs by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2014
Entry Details Article
PubMed