BDBM50429895 CHEMBL2333375

SMILES FC(F)(F)C(=O)c1ccc(cc1)C(=O)N1CCOc2ccc(cc2C1)-c1ccc2[nH]ncc2c1

InChI Key InChIKey=ZQGMPGAUEIXAHZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50429895   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Exelixis

Curated by ChEMBL

LigandBDBM50429895(CHEMBL2333375)Copy SMILESCopy InChI

Affinity DataIC50: 137nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
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