BDBM50429887 CHEMBL2332928

SMILES CS(=O)(=O)c1ccc(C(=O)N2CCOc3ccc(cc3C2)-c2ccc3nc[nH]c3c2)c(Cl)c1

InChI Key InChIKey=XVSCQIULGKNVBL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50429887   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Exelixis

Curated by ChEMBL

LigandBDBM50429887(CHEMBL2332928)Copy SMILESCopy InChI

Affinity DataIC50: 705nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate after 2 hrs by luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
9/24/2013
Entry Details Article
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