BDBM50428173 CHEMBL2336528

SMILES COc1ccc(cc1)S(=O)(=O)N(Cc1ccc(cc1)N1CCCCC1)c1ccccc1

InChI Key InChIKey=OWUYAKXOEONUBB-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50428173   

TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428173(CHEMBL2336528)
Affinity DataEC50:  49nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cell membranes assessed as inhibition of forskolin-stimulated cAMP production after 4...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428173(CHEMBL2336528)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50428173(CHEMBL2336528)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed