BDBM50420063 CHEMBL2046680

SMILES Fc1cc(ccc1Cl)C(=O)Nc1ccc(Cl)nc1

InChI Key InChIKey=JAJJZWDCPLWIET-UHFFFAOYSA-N

Data  1 IC50  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50420063   

TargetPotassium voltage-gated channel subfamily KQT member 2/3(Human)
TBA

Curated by ChEMBL

LigandBDBM50420063(CHEMBL2046680)Copy SMILESCopy InChI

Affinity DataEC50:  80nMAssay Description:Agonist activity at KCNQ2/KCNQ3 expressed in CHO cells assessed as increase in KCl-induced 86Rb+ efflux incubated for 10 mins prior to KCl-induction ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL

TargetPotassium voltage-gated channel subfamily E/KQT member 1(Human)
TBA

Curated by ChEMBL

LigandBDBM50420063(CHEMBL2046680)Copy SMILESCopy InChI

Affinity DataIC50: 1.50E+4nMAssay Description:Antagonist activity at KCNQ1/MINK expressed in CHO cells assessed as inhibition of KCl-induced 86Rb+ efflux incubated for 10 mins prior to KCl-induct...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL