BDBM50416459 CHEMBL1209347

SMILES FC(F)(F)c1ccc(Nc2nc(cs2)-c2ccccn2)cc1

InChI Key InChIKey=FEKMHFSHIMPSFV-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50416459   

TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416459(CHEMBL1209347)
Affinity DataKi:  15.8nMAssay Description:Antagonist activity at human NPY Y5 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416459(CHEMBL1209347)
Affinity DataKi:  15.8nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416459(CHEMBL1209347)
Affinity DataKi: >3.16E+4nMAssay Description:Antagonist activity at human NPY Y2 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416459(CHEMBL1209347)
Affinity DataKi: >3.16E+4nMAssay Description:Antagonist activity at human NPY Y1 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed