BDBM50401994 CHEMBL2204695

SMILES CC(C)(Oc1ccc(COc2ccc(cc2)\N=N\c2ccccc2)cc1)C(O)=O

InChI Key InChIKey=GAKQARXXOLKBGC-UHFFFAOYSA-N

Data  5 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50401994   

TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401994(CHEMBL2204695)
Affinity DataEC50:  2.10E+4nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401994(CHEMBL2204695)
Affinity DataEC50:  5.60E+3nMAssay Description:Transactivation of human GAL4-fused PPARalpha ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50401994(CHEMBL2204695)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at Gal4-fused human PPARdelta LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401994(CHEMBL2204695)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at Gal4-fused human PPARgamma LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti

Curated by ChEMBL
LigandPNGBDBM50401994(CHEMBL2204695)
Affinity DataEC50:  3.70E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalpha LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed