BDBM50401007 CHEMBL209478

SMILES CN(C)Cc1ccc(cc1)-c1ccc(CN(C)C)cc1

InChI Key InChIKey=SHOGGUIWMZFVFY-UHFFFAOYSA-N

Data  8 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50401007   

TargetHistamine H3 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-n-alpha-methylhistamine from human histamine H3 receptor homogenate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  1.32nMAssay Description:Displacement of [3H]-n-alpha-methylhistamine from human histamine H3 receptor homogenate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  1.86nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  6.61nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]-n-alpha-methylhistamine from rat histamine H3 receptor homogenate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50401007(CHEMBL209478)
Affinity DataKi:  9.33nMAssay Description:Displacement of [3H]-n-alpha-methylhistamine from rat histamine H3 receptor homogenate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed