BDBM503988 2-[[8-amino-6-(4-methylpyridin-3-yl)-2,7- naphthyridin-3-yl]amino]-6-methyl- 4H,5H,6H,7H,8H-pyrazolo[1,5- d][1,4]diazepin-7-one::US11034692, Compound 256

SMILES CN1CCc2cc(Nc3cc4cc(nc(N)c4cn3)-c3cnccc3C)nn2CC1=O

InChI Key InChIKey=QKQCFLZIFCJPTQ-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 503988   

LigandPNGBDBM503988(2-[[8-amino-6-(4-methylpyridin-3-yl)-2,7- naphthyr...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent