BDBM50396420 CHEMBL2170390

SMILES [#7]-[#6]-[#6](=O)-[#7]-[#7]-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#8])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](-[#7])=O

InChI Key InChIKey=HLJPWUIQUHGENW-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50396420   

TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)
Affinity DataEC50:  136nMAssay Description:Agonist activity at human GPR103 expressed in CHO cells co-expressing Galpha16 assessed as increase in intracellular calcium level measured for 2 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetPyroglutamylated RF-amide peptide receptor(Human)
Institute For Research and Innovation In Biomedicine (Irib)

Curated by ChEMBL
LigandPNGBDBM50396420(CHEMBL2170390)
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]26RFa from human GPR103 expressed in HEK293 cells incubated for 1 h by gamma counter based methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed