BDBM50395421 CHEMBL2165094

SMILES Cc1cc(C(N)=O)c(o1)-c1cccc(OC(=O)NCCCCCCc2ccccc2)c1

InChI Key InChIKey=FCEQLURFAJQTRC-UHFFFAOYSA-N

Data  1 KI  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50395421   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells for 5 mins by automated patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataIC50: 102nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mouse FAAH isolated from brain homogenate using [3H-ethanolamine]AEA as substrate incubated for 20 mins prior to substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataIC50: 102nMAssay Description:Inhibition of human recombinant FAAH using AMC-AA as substrate preincubated for 30 mins followed by substrate addition and measured after 30 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed
TargetFatty-acid amide hydrolase 1(Mouse)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50395421(CHEMBL2165094)
Affinity DataKi:  0.490nMAssay Description:Inhibition of mouse FAAH isolated from brain homogenate using [3H-ethanolamine]AEA as substrate incubated for 20 mins prior to substrate addition mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed