BDBM50395260 CHEMBL2163598

SMILES COc1cc(CN(C(C)C)S(=O)(=O)c2ccccn2)cc2C=CC(C)(C)Oc12

InChI Key InChIKey=LREPTZOCUMWFMS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50395260   

TargetHistone acetyltransferase p300(Human)
Emory University

Curated by ChEMBL
LigandPNGBDBM50395260(CHEMBL2163598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed