BDBM50389800 CHEMBL2070529

SMILES CCN(CC(F)F)c1ncc(cc1C)-c1cnnc2cc(OC)c(OC)cc12

InChI Key InChIKey=DBYKYMVVCSQQOF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50389800   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Amgen

Curated by ChEMBL

LigandBDBM50389800(CHEMBL2070529)Copy SMILESCopy InChI

Affinity DataIC50: 5.70nMAssay Description:Inhibition of human recombinant PDE10A using cAMP as substrate incubated for 30 mins prior to substrate addition measured after 3 hrs to overnight by...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/8/2013
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