BDBM50389597 CHEMBL2069509

SMILES C1CC(CCN1)C1N[C@H](Cc2c1[nH]c1ccccc21)c1nc(c[nH]1)-c1ccccc1

InChI Key InChIKey=RAJFOGCRMAERDF-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50389597   

TargetSomatostatin receptor type 3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50389597(CHEMBL2069509)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50389597(CHEMBL2069509)
Affinity DataIC50: 63nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
LigandPNGBDBM50389597(CHEMBL2069509)
Affinity DataIC50: 5.10E+3nMAssay Description:Displacement of [35S]MK499 from human Erg expressed in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed