BDBM50389350 CHEMBL2064100

SMILES O[C@@H]1CO[C@H]([C@H](O)[C@H]1O)c1cn(Cc2ccc(cc2)C2CC2)c2c(F)cccc12

InChI Key InChIKey=CKZTXDAVNGXTHM-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50389350   

TargetSodium/glucose cotransporter 2(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50389350(CHEMBL2064100)
Affinity DataEC50:  47nMAssay Description:Inhibition of human SGLT2 expressed in CHO-K1 cells incubated for 120 mins at 37 degC by [14C]-AMG uptake assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50389350(CHEMBL2064100)
Affinity DataEC50:  282nMAssay Description:Inhibition of human SGLT1 expressed in CHO-K1 cells incubated for 120 mins at 37 degC by [14C]-AMG uptake assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed