BDBM50382249 CHEMBL2024499

SMILES FC(F)(F)c1cc(NC(=O)Nc2cccc3ccc(NCc4ccccc4)cc23)ccc1Cl

InChI Key InChIKey=LFJKWYZEGORGJZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50382249   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Bayer Yakuhin

Curated by ChEMBL

LigandBDBM50382249(CHEMBL2024499)Copy SMILESCopy InChI

Affinity DataIC50: 140nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
2/7/2013
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