BDBM50370931 CHEMBL4162185

SMILES OC(=O)c1ccc(COc2ccc(cc2)C2C3=C(CCCC3=O)Nc3c2ccc2ccccc32)cc1

InChI Key InChIKey=OEWSFPVLNFZYKA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50370931   

TargetHistone acetyltransferase GCN5(Baker's yeast)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50370931(CHEMBL4162185)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed