BDBM50365717 CHEMBL1955990

SMILES FC(F)(F)c1cccc(c1-c1ccc2nc(C=CC3CCCCC3)[nH]c2c1)C(F)(F)F

InChI Key InChIKey=FJAIHRDKRKGFGE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50365717   

TargetTransient receptor potential M8 protein(Dog)
Janssen Pharmaceutica

Curated by ChEMBL
LigandPNGBDBM50365717(CHEMBL1955990)
Affinity DataIC50: 12.3nMAssay Description:Antagonist activity at dog TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed