BDBM50363379 CHEMBL1945882

SMILES Oc1cccc2c(O)cc(nc12)C(=O)Nc1ccccc1

InChI Key InChIKey=WCONAUUNWGJNIE-UHFFFAOYSA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50363379   

TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 74nMAssay Description:Inhibition of human plasma lipoprotein-associated phospholipase A2 using 2-thio-PAF as substrate preincubated for 20 mins measured 1 hr post substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 27nMAssay Description:Inhibition of human plasma lipoprotein-associated phospholipase A2 using 2-thio-PAF as substrate preincubated for 20 mins measured 1 hr post substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant N-terminus hexahistidine-tagged human lipoprotein-associated phospholipase A2 expressed in Escherichia coli using 2-thio-PA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant N-terminus hexahistidine-tagged human lipoprotein-associated phospholipase A2 expressed in Escherichia coli using 2-thio-PA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 270nMAssay Description:Inhibition of human plasma lipoprotein-associated phospholipase A2 using 2-thio-PAF as substrate preincubated for 20 mins measured 1 hr post substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 190nMAssay Description:Inhibition of human plasma lipoprotein-associated phospholipase A2 using 2-thio-PAF as substrate preincubated for 20 mins measured 1 hr post substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 20nMAssay Description:Inhibition of human plasma lipoprotein-associated phospholipase A2 using 2-thio-PAF as substrate preincubated for 20 mins measured 1 hr post substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 96nMAssay Description:Inhibition of recombinant N-terminus hexahistidine-tagged human lipoprotein-associated phospholipase A2 expressed in Escherichia coli using 2-thio-PA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant N-terminus hexahistidine-tagged human lipoprotein-associated phospholipase A2 expressed in Escherichia coli using 2-thio-PA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor acetylhydrolase(Human)
Activx Biosciences

Curated by ChEMBL
LigandPNGBDBM50363379(CHEMBL1945882)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant N-terminus hexahistidine-tagged, TAMRA-tagged human lipoprotein-associated phospholipase A2 expressed in Escherichia coli u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed