BDBM50362213 CHEMBL1938974

SMILES CN1C[C@H]2CN(C[C@H]2C1)C(=N)c1nc2ccc(Cl)cc2[nH]1

InChI Key InChIKey=YAAPBFJZQNGOFY-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50362213   

TargetHistamine H4 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50362213(CHEMBL1938974)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]histamine from human recombinant histamine H4 receptor expressed in CHO cells coexpressing Ga15 by radioligand filtration binding...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50362213(CHEMBL1938974)
Affinity DataKi:  56nMAssay Description:Antagonist activity at human histamine H4 receptor expressed in HEK293 cells assessed as rev inhibition of forskolin-stimulated cAMP accumulation by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed