BDBM50355916 CHEMBL1910377

SMILES Oc1ccc(cc1)-c1ccnc(c1)-c1cc2ccc(O)cc2[nH]1

InChI Key InChIKey=AXHMASICYOQTRA-UHFFFAOYSA-N

Data  2 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50355916   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Orleans University

Curated by ChEMBL

LigandBDBM50355916(CHEMBL1910377)Copy SMILESCopy InChI

Affinity DataIC50: 300nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
7/20/2012
Entry Details Article
Copy Entry DOIPubMed
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TargetCyclin-dependent kinase 5 activator 1(Human)
Orleans University

Curated by ChEMBL

LigandBDBM50355916(CHEMBL1910377)Copy SMILESCopy InChI

Affinity DataIC50: 830nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [33P-gamma]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
7/20/2012
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL