BDBM50354177 CHEMBL1836167

SMILES COC(=O)C1(CNC(=O)c2cc(OC)cc(OC)c2)CCN(Cc2ccc(cc2)C(F)(F)F)CC1

InChI Key InChIKey=ZHWCVAXYZZACNH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50354177   

TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50354177(CHEMBL1836167)
Affinity DataIC50: 4.18E+3nMAssay Description:Inhibition of T-type calcium channel alpha1G expressed in human HEK293 cells assessed as KCl-induced depolarization after 60 mins by FDSS6000 assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Korea Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50354177(CHEMBL1836167)
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed