BDBM50349877 CHEMBL1813625

SMILES CN1CCN(CC1)c1ccc(cc1)-c1cc2n(C)nc(N)c2c(=O)[nH]1

InChI Key InChIKey=VLEQHZKBZRDDGS-UHFFFAOYSA-N

Data  10 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50349877   

TargetSerine/threonine-protein kinase Chk1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of CHK1 by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of MAPKAPK2 by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetAurora kinase A(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of AurA by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibition of CK1delta by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of FYN by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of LYN by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk2(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of CHK2 by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of LCK by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of SRC by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50349877(CHEMBL1813625)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of ABL by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed