BDBM50345473 (R)-2-((R)-2-acetamido-3-phenylpropanamido)-N-((S)-1-((6S,9S,12R,13R,Z)-3-ethylidene-9-isopropyl-6,13-dimethyl-2,5,8,11-tetraoxo-1-oxa-4,7,10-triazacyclotridecan-12-ylamino)-1-oxo-3-phenylpropan-2-yl)-4-methylpentanamide::CHEMBL1784747
SMILES C\C=C1/NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](Cc2ccccc2)NC(C)=O)[C@@H](C)OC1=O)C(C)C
InChI Key InChIKey=SGGJJTTZBRPIKP-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50345473
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cell assessed as inhibition of capsaicin-induced calcium flux by fluorometric analysisMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Mouse)
University of Utah
Curated by ChEMBL
University of Utah
Curated by ChEMBL
Affinity DataIC50: 1.32E+6nMAssay Description:Antagonist activity at TRPV1 channel in C57B1 mouse dorsal root ganglion cells assessed as inhibition of capsaicin-induced calcium flux by fluorometr...More data for this Ligand-Target Pair